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Pentomone

Pentomon
Klinik ma'lumotlar

Boshqa ismlar	Lilly 113935; LY-113935
Giyohvand moddalar sinfi	Nonsteroid antiandrogen
ATC kodi	Yo'q
Identifikatorlar
IUPAC nomi (5aS, 6aR, 12aS, 13aR) -4,8-dimetoksi-6,6-dimetil-5a, 6a, 12,12a, 13a, 14-geksahidroxromeno [3,2-b] ksanten-13-bir
CAS raqami	67102-87-8
PubChem CID	49354
ChemSpider	44862
UNII	OPS67T329P
ChEMBL	ChEMBL2107005
Kimyoviy va fizik ma'lumotlar
Formula	C₂₄H₂₆O₅
Molyar massa	394.467 g · mol⁻¹
3D model (JSmol)	Interaktiv rasm
Jilmayganlar CC1 (C2C (CC3 = C (O2) C (= CC = C3) OC) C (= O) C4C1OC5 = C (C4) C = CC = C5OC) C
InChI InChI = InChI = 1S / C24H26O5 / c1-24 (2) 22-15 (11-13-7-5-9-17 (26-3) 20 (13) 28-22) 19 (25) 16-12- 14-8-6-10-18 (27-4) 21 (14) 29-23 (16) 24 / h5-10,15-16,22-23H, 11-12H2,1-4H3 / t15-, 16 +, 22-, 23 + Kalit: MTJTVTZUEKVNTG-YJEDKTMASA-N

Pentomon (KARVONSAROY, USAN) (rivojlanish kodining nomi Lilly 113935 yoki LY-113935) a steroid bo'lmagan antiandrogen (NSAA) "deb ta'riflanganprostata o'sish inhibitori "bu hech qachon bozorga chiqarilmagan.^[1] U 1978 yilda sintez qilingan va tahlil qilingan.^[1]

Adabiyotlar

^ ^a ^b Elks J (2014 yil 14-noyabr). Dori vositalari lug'ati: kimyoviy ma'lumotlar: kimyoviy ma'lumotlar, tuzilmalar va bibliografiyalar. Springer. 949– betlar. ISBN 978-1-4757-2085-3.

Androgen retseptorlari modulyatorlar

Agonistlar	Testosteron hosilalari: 4-Androstenediol 4-dehidroepiandrosteron (4-DHEA) 4-gidroksitestosteron 4,17a-dimetiltestosteron 5-Androstenedion 11-ketotestosteron 11β-gidroksiandrostenedion Adrenosteron (11-ketoandrostenedion, 11-oksoandrostenedion) Androstenediol (5-androstenediol) Androstenediol 3β-asetat Androstenediol 17β-asetat Androstenediol diatsetat Androstenediol dipropionat Androstenedion (4-androstenedion) Atamestane Boldenone Boldenone undesilenat Boldion (1,4-androstadienedion) Klostebol Klostebol asetat Clostebol kaproati Clostebol propionat Kloksotestosteron Kloksotestosteron asetat Dehidroandrosteron DHEA (androstenolon, prasteron; 5-DHEA) DHEA enanthate (prasterone enanthate) DHEA sulfat Exemestane Formestan Plomestane Quinbolone Silandrone Testosteron^# (+ dutasterid) Testosteron efirlari Polytestosterone phloretin fosfat 5a-Dihidrotestosteron hosilalari: 1-Androstenediol 1-Androstenedion 1-Androsteron (1-andro, 1-DHEA) 1-testosteron 3a-Androstandiol 5a-Androst-2-en-17-one 7β-gidroksiepiandrosteron 11-ketodihidrotestosteron Androsteron Bolazin Bolazin kapronat Dihidroetiltestosteron Dihidrofluoksimesteron Dihidrometilandrostenediol Dihidrotestosteron (DHT) (androstanolon, stanolon) Dihidrotestosteron esterlari Drostanolon Drostanolon propionat Epiandrosteron Epitiostanol Mepitiostane Mesabolone Mesterolon Mesterolon sipionat Metildiazinol Nisterime Nisterim asetat Prostanozol Stenbolone Stenbolon asetat Guvohnoma (testiphenon, testiphenone) 19-Nortestosteron hosilalari: 7a-Metil-19-norandrostenedion (MENT dione, trestione) 11β-Metil-19-nortestosteron 11β-Metil-19-nortestosteron dodesilkarbonat 19-Nor-5-androstenediol 19-Nor-5-androstenedion 19-Nordehidroepiandrosteron Bolandiol Bolandiol dipropionat Bolandione (19-nor-4-androstenedione) Bolmantalat (nandrolone adamantoate) Dienedione Dienolon Dimetandrolon Dimetandrolon bükiklat Dimetandrolon dodesilkarbonat Dimethandrolone undecanoate LS-1727 (nandrolon 17β-N- (2-xloretil) -N-nitrosokarbamat) Metoksidiyenon (metoksigonadien) Nandrolone Nandrolon esterlari Norklostebol Norklostebol asetat Normetandron (metilestrenolon, normetisteron) Oksabolone Oksabolon sipionat (oksabolon kipionat) Trenbolone Trenbolone asetat Trenbolone enanthate Trenbolone geksahidrobenzilkarbonat Trenbolone undecanoate Trendione Trestolon (MENT) Trestolon asetat Trestolon enantati 5a-Dihidro-19-nortestosteron hosilalari: 5a-Dihidronandrolon 5a-Dihidrotrestolon 19-Norandrosteron 17a-alkillangan testosteron hosilalari: Bolasterone Kalusteron Xlorodehidrometilandrostenediol (CDMA) Xlorodehidrometiltestosteron (CDMT) Xlorometilandrostenediol (CMA) Enestebol Etilestosteron Fluoksimesteron Formebolone Gidroksistenozol Metandienone (metandrostenolon) Metandriol (metilandrostenediol) Metandriol bisenantoil asetat Metandriol diatsetat Metandriol dipropionat Metandriol propionat Metilklostebol (xlorometiltestosteron) Metiltestosteron (+ esterlangan estrogenlar) Metiltestosteron 3-heksil efir Oksimesteron Penmesterol Tiomesteron 17a-alkillangan 5a-dihidrotestosteron hosilalari: Androizoksazol Desoksimetiltestosteron Furazabol Mebolazin (dimetazin) Mestanolone Metenolon Metenolon asetat Metenolon enantat Metasteron Metil-1-testosteron Metilepitiostanol Metilstenbolon Oxandrolone Oksimetolon Stanozolol 17a-alkilatlangan 19-nortestosteron hosilalari: Bolenol Dimetildienolon Dimetiltrienolon Etildienolon Etilestrenol Metildienolon Metilhidroksinandrolon (MOHN, MHN) Metribolon Miboleron Norboleton Noretandrolon Propetandrol RU-2309 Tetrahidrogestrinon 17a-alkillangan 5a-dihidro-19-nortestosteron hosilalari: 5a-Dihidronoretandrolon 5a-Dihidronormetandron 17a-Viniltestosteron hosilalari: Norvinisteron (vinilnortestosteron) 17a-Vinil-19-nortestosteron hosilalari: Viniltestosteron 17a-etiniltestosteron hosilalari: Danazol Etinilendrostenediol Etandrostat Etisteron (etiniltestosteron) 5a-Dihidro-17a-etiniltestosteron hosilalari: 17a-etinil-3a-androstandiol 17a-etinil-3b-androstandiol Dihidroetisteron 17a-etinil-19-nortestosteron hosilalari: Δ⁴-Tibolon Desogestrel Etonogestrel Etinodiol Etinodiol diatsetat Gestoden Gestrinone Levonorgestrel Levonorgestrel esterlari (masalan, levonorgestrel butanoat) Lynestrenol Lynestrenol fenilpropionat Noretisteron Noretisteron esterlari (masalan, noretisteron asetat, norethisterone enanthate) Norgestrel Norgestrienon Quingestanol Quingestanol asetat Tibolone 5a-Dihidro-17a-etinil-19-nortestosteron hosilalari: 5a-Dihidrolevonorgestrel 5a-Dihidronorististeron Progesteron hosilalari: 6a-metilprogesteron Medroksiprogesteron asetat Megestrol asetat Boshqalar / saralanmagan: 3-Keto-5a-abirateron 5a-Androstan Alternariyol Cl-4AS-1 Drupanol Trilostan ZM-182345
Aralashgan (SARMlar)	Nonsteroidal: 198RL26 ACP-105 AC-262536 Asetotiolutamid Andarin (asetamidoksolutamid, androksolutamid, GTx-007, S-4) BMS-564929 DTIB Enobosarm (ostarin, MK-2866, GTx-024, S-22) FTBU-1 GSK2881078 GSK-4336A GSK-8698 LG-121071 (LGD-121071) LGD-2226 LGD-2941 (LGD-122941) LGD-3303 LGD-4033 LY-2452473 JNJ-26146900 JNJ-28330835 JNJ-37654032 ORM-11984 R-1 RAD140 RU-59063 S-1 S-23 S-40503 S-101479 Triklosan Steroidal: EM-9017 MK-0773 TFM-4AS-1 YK-11
Antagonistlar	Steroidal: 7a-tioprogesteron 7a-tiospironolakton 7a-tiometilspironolakton 11a-gidroksiprogesteron 15β-gidroksitsiproteron asetat Abiraterone Abirateron asetat Allitestosteron Benorterone BOMT Kanrenoik kislota Kanrenon Xlormadinon asetat Klasoteron Klometeron Siproheptadin Kiproteron Siproteron asetat Delanteron Delmadinon asetat Dicirenone Dienogest Drospirenone DU-41165 Edogestrone EM-4350 EM-5854 EM-5855 EM-6537 Epitestosteron Galeterone Guggulsterone Ludaterone Medrogestone Megestrol asetat Mespirenone Metogest Mexrenone Mifepriston Nomegestrol asetat Nordinone Osaterone Osateron asetat Oksendolon Kaliy canrenoate Promegestone Prorenone Rosterolon RU-15328 SC-5233 (spirolakton) Spironolakton Spirorone Spiroksazon Topteron Trimegestone Trimetiltrienolon (R-2956) Zanoterone Nonsteroidal: 5N-Bikalutamid AA560 Antarklidlar Arabilin Apalutamid Atrarik kislota AZD-3514 Bakuchiol BAY-1024767 Bikalutamid Bisfenollar (masalan, BADGE, BFDGE, bisfenol A, bisfenol F, bisfenol S) BMS-501949 BMS-570511 BMS-641988 CH5137291 Simetidin Cioteronel Siyanilutamid Darolutamid DDT (metabolit orqali p, p’-DDE) Dildrin DIMP Endosulfan Enzalutamid EPI-001 EPI-7386 Fenarimol Flutamid Gidroksiflutamid Inokoteron Inokoteron asetat Ketokonazol Ketodarolutamid Lavanda yog'i LG-105 LG-120907 LGD-1331 Linuron Metiokarb N-Butilbenzensulfonamid N-Desmetilapalutamid N-Desmetilenzalutamid Nilutamid ONC1-13B Pentomon PF-998425 Fenotrin Proxloraz Prokimidon Proksalutamid Ralaniten (EPI-002) Ralaniten atsetat (EPI-506) RD-162 Rezvilutamid Ro 2-7239 Ro 5-2537 RU-22930 RU-56187 RU-57073 RU-58642 RU-58841 Seviteronel Talidomid Topilutamid (fluridil) Valproik kislota Vinclozolin YM-580 YM-92088 YM-175735

GPRC6A

Agonistlar	Kationlar (shu jumladan) alyuminiy, kaltsiy, gadoliniy, magniy, stronsiyum, rux) Dehidroandrosteron Dihidrotestosteron Estradiol L-a-aminokislotalar (shu jumladan) L- arginin, L-lisin, L-ornitin) Osteokalsin SHBG Testosteron

Shuningdek qarang: Retseptor / signalizatsiya modulyatorlari; Androgenlar va antiandrogenlar; Estrogen retseptorlari modulyatorlari; Progesteron retseptorlari modulyatorlari; Androgenlar / anabolik steroidlar ro'yxati

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