| 
|---|
| 5-HT1 | | 5-HT1A | - Agonistlar: 8-OH-DPAT
 - Adatanserin
 - Amfetamin
 - Antidepressantlar (masalan, etoperidon, gidroksifazodon, nefazodon, trazodon, triazoledion, vilazodon, vortioksetin)
 - Atipik antipsikotiklar (masalan, aripiprazol, asenapin, brekspiprazol, kariprazin, klozapin, lurasidon, ketiapin, ziprasidon)
 - Azapironlar (masalan, buspirone, eptapiron, gepiron, perospiron, tandospiron)
 - Bay R 1531
 - Befiradol
 - BMY-14802
 - Kannabidiol
 - Dimemebfe
 - Dopamin
 - Ebalzotan
 - Eltoprazin
 - Entsiprazin
 - Ergolines (masalan, bromokriptin, kabergolin, dihidroergotamin, ergotamin, lisurid, LSD, metilergometrin (metlergonovin), metizergid, pergolit)
 - F-11461
 - F-12826
 - F-13714
 - F-14679
 - F-15063
 - F-15,599
 - Flesinoksan
 - Flibanserin
 - Flumeksadol
 - Lesopitron
 - LY-293284
 - LY-301317
 - mCPP
 - MKC-242
 - Naluzotan
 - NBUMP
 - Osemozotan
 - Oksaflozan
 - Pardoprunoks
 - Piklozotan
 - Rawolscine
 - Repinotan
 - Roksindol
 - RU-24,969
 - S-14506
 - FZR 14671
 - FZR-15535
 - Sarizotan
 - Serotonin (5-HT)
 - SSR-181507
 - Sunepitron
 - Triptaminlar (masalan, 5-CT, 5-MeO-DMT, 5-MT, bufotenin, DMT, o'zlashtirmoq, N-Me-5-HT, psilotsin, psilotsibin)
 - TGBA01AD
 - U-92,016-A
 - Urapidil
 - Vilazodone
 - Xaliproden
 - Yohimbine
 
  |  - Antagonistlar: Atipik antipsikotiklar (masalan, iloperidon, risperidon, sertindol)
 - AV965
 - Beta blokerlar (masalan, alprenolol, karteolol, siyanopindolol, yodosiyanopindolol, izamoltan, oksprenolol, penbutolol, pindobind, pindolol, propranolol, tertatolol)
 - BMY-7,378
 - CSP-2503
 - Dotarizin
 - Ergolines (masalan, metrgolin)
 - FCE-24379
 - Flopropion
 - GR-46611
 - Isamoltan
 - Lekozotan
 - Mefway
 - Metitepin (metiotepin)
 - MIN-117 (WF-516)
 - MPPF
 - NAN-190
 - Robalzotan
 - FZR-15535
 - SB-649,915
 - SDZ 216-525
 - Spiperon
 - Spiramid
 - Spiroksatrin
 - UH-301
 - YO'L-100135
 - YO'L-100635
 - Ksilamidin
 
  |   |  
  | 
|---|
 | 5-HT1B | - Agonistlar: CGS-12066A
 - CP-93129
 - CP-94253
 - CP-122,288
 - CP-135807
 - Eltoprazin
 - Ergolines (masalan, bromokriptin, dihidroergotamin, ergotamin, metilergometrin (metlergonovin), metizergid, pergolit)
 - mCPP
 - RU-24,969
 - Serotonin (5-HT)
 - Triptanlar (masalan, avitriptan, donitriptan, eletriptan, sumatriptan, zolmitriptan)
 - TFMPP
 - Triptaminlar (masalan, 5-BT, 5-CT, 5-MT, DMT)
 - Vortioksetin
 
  |   |   |  
  | 
|---|
 | 5-HT1D | - Agonistlar: CP-122,288
 - CP-135807
 - CP-286601
 - Ergolines (masalan, bromokriptin, kabergolin, dihidroergotamin, ergotamin, LSD, metizergid)
 - GR-46611
 - L-694247
 - L-772405
 - mCPP
 - PNU-109291
 - PNU-142633
 - Serotonin (5-HT)
 - TGBA01AD
 - Triptanlar (masalan, almotriptan, avitriptan, donitriptan, eletriptan, frovatriptan, naratriptan, rizatriptan, sumatriptan, zolmitriptan)
 - Triptaminlar (masalan, 5-BT, 5-CT, 5-Et-DMT, 5-MT, 5- (noniloksi) triptamin, DMT)
 
  |   |   |  
  | 
|---|
 | 5-HT1E |  | 
|---|
 | 5-HT1F |  | 
|---|
 
  | 
|---|
| 5-HT2 | | 5-HT2A | - Agonistlar: 25H / NB seriyali (masalan, 25I-NBF, 25I-NBMD, 25I-NBOH, 25I-NBOMe, 25B-NBOMe, 25C-NBOMe, 25TFM-NBOMe, 2CBCB-NBOMe, 25CN-NBOH, 2CBFly-NBOMe)
 - 2C (masalan, 2C-B, 2C-E, 2C-I, 2C-T-2, 2C-T-7, 2C-T-21)
 - 2C-B-FLY
 - 2CB-ind
 - 5-metoksitriptaminlar (5-MeO-DET, 5-MeO-DiPT, 5-MeO-DMT, 5-MeO-DPT, 5-MT)
 - a-alkilriptaminlar (masalan, 5-Cl-aMT, 5-Fl-aMT, 5-MeO-aET, 5-MeO-aMT, a-Me-5-HT, aET, aMT)
 - AL-34662
 - AL-37350A
 - Bromo-DragonFLY
 - Dimemebfe
 - DMBMPP
 - DOx (masalan, DOB, DOC, DOI, DOM)
 - Efavirenz
 - Ergolines (masalan, 1P-LSD, ALD-52, bromokriptin, kabergolin, ergine (LSA), ergometrin (ergonovin), ergotamin, lisurid, LA-SS-Az, LSB, LSD, LSD-Pip, LSH, LSP, metilergometrin (metlergonovin), pergolit)
 - Flumeksadol
 - Jimkalin
 - Lorcaserin
 - MDxx (masalan, MDA (tenamfetamin), MDMA (midomafetamin), MDOH, MMDA)
 - O-4310
 - Oksaflozan
 - PHA-57378
 - PNU-22394
 - PNU-181731
 - RH-34
 - Fenetilaminlar (masalan, lofofin, meskalin)
 - Piperazinlar (masalan, BZP, quipazin, TFMPP)
 - Serotonin (5-HT)
 - TCB-2
 - TFMFly
 - Triptaminlar (masalan, 5-BT, 5-CT, bufotenin, DET, DiPT, DMT, DPT, psilotsin, psilotsibin, triptamin)
 
  |  - Antagonistlar: 5-I-R91150
 - 5-MeO-NBpBrT
 - AC-90179
 - Adatanserin
 - Altanserin
 - Antihistaminiklar (masalan, siproheptadin, gidroksin, ketotifen, perlapin)
 - AMDA
 - Atipik antipsikotiklar (masalan, amperozid, aripiprazol, asenapin, blonanserin, brekspiprazol, karpipramin, klokapramin, klorotepin, klozapin, fluperlapin, gevotrolin, iloperidon, lurasidon, melperone, mosapramin, okaperidon, olanzapin, paliperidon, ketiapin, risperidon, sertindol, zikronapin, ziprasidon, zotepin)
 - Cinanserin
 - CSP-2503
 - Deramciclane
 - Dotarizin
 - Eplivanserin
 - Ergolines (masalan, amergid, LY-53857, LY-215,840, mezulerjin, metrgolin, metizergid, sergoleksol)
 - Fananserin
 - Flibanserin
 - Glemanserin
 - Irindalone
 - Ketanserin
 - KML-010
 - Landipirdin
 - LY-393558
 - mCPP
 - Medifoksamin
 - Metitepin (metiotepin)
 - MIN-117 (WF-516)
 - Naftidrofuril
 - Nantenin
 - Nelotanserin
 - Opiranserin (VVZ-149)
 - Pelanserin
 - Fenoksibenzamin
 - Pimavanserin
 - Pirenperone
 - Pizotifen
 - Pruvanserin
 - Rawolscine
 - Ritanserin
 - Roluperidon
 - FZR 14671
 - Sarpogrelate
 - Serotonin antagonistlari va qaytarib olish inhibitörleri (masalan, etoperidon, gidroksifazodon, lubazodon, mepiprazol, nefazodon, triazoledion, trazodon)
 - SR-46349B
 - TGBA01AD
 - Teniloksazin
 - Temanogrel
 - Tetratsiklik antidepressantlar (masalan, amoksapin, aptazapin, esmirtazapin, maprotilin, mianserin, mirtazapin)
 - Trisiklik antidepressantlar (masalan, amitriptilin)
 - Odatda antipsikotiklar (masalan, xlorpromazin, flüfenazin, haloperidol, loxapin, perfenazin, pimozid, pipamperon, proxlorperazin, setoperon, spiperon, spiramid, tioridazin, tiyotiksen, trifluoperazin)
 - Volinanserin
 - Ksilamidin
 - Yohimbine
 
  |   |  
  | 
|---|
 | 5-HT2B | - Agonistlar: 4-metilaminoreks
 - Aminorex
 - Amfetaminlar (masalan, xlorfentermin, cloforex, dexfenfluramin, fenfluramin, levofenfluramin, norfenfluramin)
 - BW-723C86
 - DOx (masalan, DOB, DOC, DOI, DOM)
 - Ergolines (masalan, kabergolin, dihidroergokriptin, dihidroergotamin, ergotamin, metilergometrin (metlergonovin), metizergid, pergolit)
 - Lorcaserin
 - MDxx (masalan, MDA (tenamfetamin), MDMA (midomafetamin), MDOH, [MMDA (dori)
 
  |  - Antagonistlar: Agomelatin
 - Atipik antipsikotiklar (masalan, amisulprid, aripiprazol, asenapin, brekspiprazol, kariprazin, klozapin, N-desalkilquetiapin (norquetiapin), N-desmetilklozapin (norklozapin), olanzapin, pipamperon, ketiapin, risperidon, ziprasidon)
 - Siproheptadin
 - EGIS-7625
 - Ergolines (masalan, amergid, bromokriptin, lisurid, LY-53857, LY-272015, mezulerjin)
 - Ketanserin
 - LY-393558
 - mCPP
 - Metadoksin
 - Metitepin (metiotepin)
 - Pirenperone
 - Pizotifen
 - Propranolol
 - PRX-08066
 - Rawolscine
 - Ritanserin
 - RS-127445
 - Sarpogrelate
 - SB-200646
 - SB-204741
 - SB-206553
 - SB-215505
 - SB-221284
 - SB-228357
 - SDZ SER-082
 - Tegaserod
 - Tetratsiklik antidepressantlar (masalan, amoksapin, mianserin, mirtazapin)
 - Trazodone
 - Odatda antipsikotiklar (masalan, xlorpromazin)
 - TIK-301
 - Yohimbine
 
  |   |  
  | 
|---|
 | 5-HT2C | - Agonistlar: 2C (masalan, 2C-B, 2C-E, 2C-I, 2C-T-2, 2C-T-7, 2C-T-21)
 - 5-metoksitriptaminlar (5-MeO-DET, 5-MeO-DiPT, 5-MeO-DMT, 5-MeO-DPT, 5-MT)
 - a-alkilriptaminlar (masalan, 5-Cl-aMT, 5-Fl-aMT, 5-MeO-aET, 5-MeO-aMT, a-Me-5-HT, aET, aMT)
 - A-372159
 - AL-38022A
 - Alstonin
 - CP-809101
 - Dimemebfe
 - DOx (masalan, DOB, DOC, DOI, DOM)
 - Ergolines (masalan, ALD-52, kabergolin, dihidroergotamin, ergine (LSA), ergotamin, lisurid, LA-SS-Az, LSB, LSD, LSD-Pip, LSH, LSP, pergolit)
 - Flumeksadol
 - Lorcaserin
 - MDxx (masalan, MDA (tenamfetamin), MDMA (midomafetamin), MDOH, MMDA)
 - MK-212
 - ORG-12962
 - ORG-37684
 - Oksaflozan
 - PHA-57378
 - Fenetilaminlar (masalan, lofofin, meskalin)
 - Piperazinlar (masalan, aripiprazol, BZP, mCPP, quipazin, TFMPP)
 - PNU-22394
 - PNU-181731
 - Ro60-0175
 - Ro60-0213
 - Serotonin (5-HT)
 - Triptaminlar (masalan, 5-BT, 5-CT, bufotenin, DET, DiPT, DMT, DPT, psilotsin, psilotsibin, triptamin)
 - Vabikaserin
 - YO'L-629
 - YO'L-161503
 - YM-348
 
  |  - Antagonistlar: Adatanserin
 - Agomelatin
 - Atipik antipsikotiklar (masalan, asenapin, klorotepin, klozapin, fluperlapin, iloperidon, melperone, olanzapin, paliperidon, ketiapin, risperidon, sertindol, ziprasidon, zotepin)
 - Captodiame
 - CEPC
 - Cinanserin
 - Siproheptadin
 - Deramciclane
 - Desmetramadol
 - Dotarizin
 - Eltoprazin
 - Ergolines (masalan, amergid, bromokriptin, LY-53857, LY-215,840, mezulerjin, metrgolin, metizergid, sergoleksol)
 - Etoperidon
 - Fluoksetin
 - FR-260010
 - Irindalone
 - Ketanserin
 - Ketotifen
 - Latrepirdin (dimebolin)
 - Medifoksamin
 - Metitepin (metiotepin)
 - Nefazodon
 - Pirenperone
 - Pizotifen
 - Propranolol
 - Ritanserin
 - RS-102221
 - FZR 14671
 - SB-200646
 - SB-206553
 - SB-221284
 - SB-228357
 - SB-242084
 - SB-243213
 - SDZ SER-082
 - Tedatioksetin
 - Tetratsiklik antidepressantlar (masalan, amoksapin, aptazapin, esmirtazapin, maprotilin, mianserin, mirtazapin)
 - TIK-301
 - Tramadol
 - Trazodone
 - Trisiklik antidepressantlar (masalan, amitriptilin, nortriptilin)
 - Odatda antipsikotiklar (masalan, xlorpromazin, loxapin, pimozid, pipamperon, tioridazin)
 - Ksilamidin
 
  |   |  
  | 
|---|
 
  | 
|---|
| 5-HT3–7 | | 5-HT3 | - Agonistlar: Spirtli ichimliklar (masalan, butanol, etanol (alkogol), trikloroetanol)
 - m-CPBG
 - Fenilbiguanid
 - Piperazinlar (masalan, BZP, mCPP, quipazin)
 - RS-56812
 - Serotonin (5-HT)
 - SR-57227
 - SR-57227A
 - Triptaminlar (masalan, 2-Me-5-HT, 5-CT, bufotenidin (5-HTQ))
 - Uchuvchi moddalar / gazlar (masalan, halotan, izofluran, toluol, trikloretan)
 - YM-31636
 
  |  - Antagonistlar: Alosetron
 - Arazasetron
 - AS-8112
 - Atipik antipsikotiklar (masalan, klozapin, olanzapin, ketiapin)
 - Azasetron
 - Batanoprid
 - Bemesetron (MDL-72222)
 - Bupropion
 - Cilansetron
 - CSP-2503
 - Dazoprid
 - Dolasetron
 - Galanolakton
 - Granisetron
 - Gidroksibupropion
 - ICS-205930
 - Lerisetron
 - Memantin
 - Ondansetron
 - Palonosetron
 - Ramosetron
 - Renzaprid
 - Rikasetron
 - Tedatioksetin
 - Tetratsiklik antidepressantlar (masalan, amoksapin, mianserin, mirtazapin)
 - Thujone
 - Tropanserin
 - Tropisetron
 - Odatda antipsikotiklar (masalan, loxapin)
 - Uchuvchi moddalar / gazlar (masalan, azot oksidi, sevofluran, ksenon)
 - Vortioksetin
 - Zakoprid
 - Zatosetron
 
  |   |  
  | 
|---|
 | 5-HT4 |  | 
|---|
 | 5-HT5A |  | 
|---|
 | 5-HT6 | - Agonistlar: Ergolines (masalan, dihidroergokriptin, dihidroergotamin, ergotamin, lisurid, LSD, mezulerjin, metrgolin, metizergid)
 - Serotonin (5-HT)
 - Triptaminlar (masalan, 2-Me-5-HT, 5-BT, 5-CT, 5-MT, Bufotenin, E-6801, E-6837, EMD-386088, EMDT, LY-586713, N-Me-5-HT, triptamin)
 - YO'L-181187
 - YO'L-208466
 
  |  - Antagonistlar: ABT-354
 - Atipik antipsikotiklar (masalan, aripiprazol, asenapin, klorotepin, klozapin, fluperlapin, iloperidon, olanzapin, tiospiron)
 - AVN-101
 - AVN-211
 - AVN-322
 - AVN-397
 - BGC20-760
 - BVT-5182
 - BVT-74316
 - Cerlapirdin
 - EGIS-12,233
 - GW-742457
 - Idalopirdin
 - Ketanserin
 - Landipirdin
 - Latrepirdin (dimebolin)
 - Masupirdin
 - Metitepin (metiotepin)
 - MS-245
 - PRX-07034
 - Ritanserin
 - Ro 04-6790
 - Ro 63-0563
 - SB-258585
 - SB-271046
 - SB-357134
 - SB-399885
 - SB-742457
 - Tetratsiklik antidepressantlar (masalan, amoksapin, mianserin)
 - Trisiklik antidepressantlar (masalan, amitriptilin, klomipramin, doksepin, nortriptilin)
 - Odatda antipsikotiklar (masalan, xlorpromazin, loxapin)
 
  |   |  
  | 
|---|
 | 5-HT7 |  |  - Antagonistlar: Atipik antipsikotiklar (masalan, amisulprid, aripiprazol, asenapin, brekspiprazol, klorotepin, klozapin, fluperlapin, olanzapin, risperidon, sertindol, tiospiron, ziprasidon, zotepin)
 - Butaklamol
 - DR-4485
 - EGIS-12,233
 - Ergolines (masalan, 2-Br-LSD (BOL-148), amergid, bromokriptin, kabergolin, dihidroergotamin, ergotamin, LY-53857, LY-215,840, mezulerjin, metrgolin, metizergid, sergoleksol)
 - JNJ-18038683
 - Ketanserin
 - LY-215,840
 - Metitepin (metiotepin)
 - Ritanserin
 - SB-258719
 - SB-258741
 - SB-269970
 - SB-656104
 - SB-656104A
 - SB-691673
 - SLV-313
 - SLV-314
 - Spiperon
 - SSR-181507
 - Tetratsiklik antidepressantlar (masalan, amoksapin, maprotilin, mianserin, mirtazapin)
 - Trisiklik antidepressantlar (masalan, amitriptilin, klomipramin, imipramin)
 - Odatda antipsikotiklar (masalan, asetofenazin, xlorpromazin, xlorprotiksen, flüfenazin, loxapin, pimozid)
 - Vortioksetin
 
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